Ingredient Details :Olibanumol B


TCMI-ID: TCMI18090


Physicochemical Property
Ingredient Name Olibanumol B
Pubchem CID 44233147
Iupac name (1S,2S,3R,5S)-2-methyl-5-propan-2-ylbicyclo[3.1.0]hexane-2,3-diol
Molecular Formula C10H18O2
Molecular Weight 170.25
Isomeric smiles CC(C)[C@@]12C[C@@H]1[C@]([C@@H](C2)O)(C)O
InChI InChI=1S/C10H18O2/c1-6(2)10-4-7(10)9(3,12)8(11)5-10/h6-8,11-12H,4-5H2,1-3H3/t7-,8-,9+,10+/m1/s1
InChIKey PRHLXOXJZCCENK-IMSYWVGJSA-N
External Database Links HERB2.0: HBIN038059   TCMSID: 1255  
Structural Information
nHA(Number of hydrogen bond acceptors) 2
nHD(Number of hydrogen bond donors) 2
nRot(Number of rotatable bonds) 1
nRing(Number of rings) 2
MaxRing(Number of atoms in the biggest ring) 6
nHet(Number of heteroatoms) 2

Stability
nRig(Number of rigid bonds) 7
Flexibility 0.143
Stereo Centers(Number of stereocenters) 4

Solubility
TPSA(Topological polar surface area) 40.46
logS(The logarithm of aqueous solubility value) -1.144
logP(The logarithm of the n-octanol/water distribution coefficient) 1.529
logD7.4(The logarithm of the n-octanol/water distribution coefficients at pH=7.4) 0.85

Pharmacokinetic Property
Quantitative Estimate of Drug-likeness 0.62
Synthetic accessibility score 4.453
Natural Product-likeness score 3.096
Lipinski Rule Accepted
GSK Rule Accepted
Golden Triangle Rejected

Absorption
Caco-2 Permeability -4.68
MDCK Permeability 1.68E-05
Pgp-substrate 0.6
HIA(human intestinal absorption) 0.005
F20%(20% Oral Bioavailability) 0.006
F30%(30% Oral Bioavailability) 0.129

Distribution
PPB(Plasma protein binding) 54.70%
VD(Volume Distribution) 1.442
BBB Penetration(Blood brain barrier penetration) 0.828
B3 Penetration(Blood brain barrier penetration) Permeable
Fu(The fraction unbound in plasms) 55.52%

Metabolism
CYP1A2 inhibitor 0.047
CYP1A2 substrate 0.373
CYP2C19 inhibitor 0.02
CYP2C19 substrate 0.809
CYP2C9 inhibitor 0.015
CYP2C9 substrate 0.13
CYP2D6 inhibitor 0.006
CYP2D6 substrate 0.26
CYP3A4 inhibitor 0.129
CYP3A4 substrate 0.236

Excretion
CL(The clearance of a drug) 8.345
T1/2 0.516

Toxicology
NonBiodegradable Rule 0
Pfizer Rule Accepted
SR-MMP 0.099

Toxic Dose
FDAMDD(FDA Maximum (Recommended) Daily Dose) 0.147
IGC50 2.088
LC50FM 2.387
LC50DM 3.205

Reproductive Effects
NR-AR(Androgen receptor) 0.535
NR-AR-LBD(Androgen receptor) 0.026
NR-Aromatase 0.012
NR-ER(Estrogen receptor) 0.152
NR-ER-LBD(Estrogen receptor) 0.015

Allergy
Skin Sensitization Rule 0
Skin Sensitization 0.318

Acute Toxicity
Acute Toxicity Rule 1
Rat Oral Acute Toxicity 0.847

Organ Toxicity
hERG Blockers 0.031
H-HT(The human hepatotoxicity) 0.417
DILI(Drug-induced liver injury) 0.044

Primary Irritation
Eye Corrosion 0.575
Eye Irritation 0.955
Respiratory Toxicity 0.961

Mutagenic Effects
AMES Toxicity 0.018

Tumorigenic Effects
Carcinogencity 0.732
SR-ARE(Antioxidant Response Element) 0.026
SR-ATAD5(ATPase family AAA domain-containing protein 5) 0.016
SR-p53 0.017

Related TCM-Disorder Names

Related Formulae

Related Herbs

Related Targets

Network Analysis

Copyright © Chengdu University of TCM All rights reserved.