Ingredient Details :3-Methylcyclopropene


TCMI-ID: TCMI07369


Physicochemical Property
Ingredient Name 3-Methylcyclopropene
Pubchem CID 638076
Iupac name 3-methylcyclopropene
Molecular Formula C4H6
Molecular Weight 54.09
Isomeric smiles CC1C=C1
InChI InChI=1S/C4H6/c1-4-2-3-4/h2-4H,1H3
InChIKey FAPGNCCCFGCZKP-UHFFFAOYSA-N
External Database Links TCMSuite: 43634  
Structural Information
nHA(Number of hydrogen bond acceptors) 0
nHD(Number of hydrogen bond donors) 0
nRot(Number of rotatable bonds) 0
nRing(Number of rings) 1
MaxRing(Number of atoms in the biggest ring) 3
nHet(Number of heteroatoms) 0

Stability
nRig(Number of rigid bonds) 3
Flexibility 0
Stereo Centers(Number of stereocenters) 0

Solubility
TPSA(Topological polar surface area) 0
logS(The logarithm of aqueous solubility value) -0.92
logP(The logarithm of the n-octanol/water distribution coefficient) 1.775
logD7.4(The logarithm of the n-octanol/water distribution coefficients at pH=7.4) 1.356

Pharmacokinetic Property
Quantitative Estimate of Drug-likeness 0.364
Synthetic accessibility score 2.638
Natural Product-likeness score 1.03
Lipinski Rule Accepted
GSK Rule Accepted
Golden Triangle Rejected

Absorption
Caco-2 Permeability -4.186
MDCK Permeability 3.73E-05
Pgp-substrate 0.004
HIA(human intestinal absorption) 0.004
F20%(20% Oral Bioavailability) 0.001
F30%(30% Oral Bioavailability) 0.077

Distribution
PPB(Plasma protein binding) 64.71%
VD(Volume Distribution) 1.639
BBB Penetration(Blood brain barrier penetration) 0.989
B3 Penetration(Blood brain barrier penetration) Permeable
Fu(The fraction unbound in plasms) 44.17%

Metabolism
CYP1A2 inhibitor 0.776
CYP1A2 substrate 0.848
CYP2C19 inhibitor 0.117
CYP2C19 substrate 0.856
CYP2C9 inhibitor 0.025
CYP2C9 substrate 0.407
CYP2D6 inhibitor 0.03
CYP2D6 substrate 0.442
CYP3A4 inhibitor 0.115
CYP3A4 substrate 0.225

Excretion
CL(The clearance of a drug) 8.435
T1/2 0.649

Toxicology
NonBiodegradable Rule 0
Pfizer Rule Accepted
SR-MMP 0.007

Toxic Dose
FDAMDD(FDA Maximum (Recommended) Daily Dose) 0.043
IGC50 2.608
LC50FM 3.63
LC50DM 3.794

Reproductive Effects
NR-AR(Androgen receptor) 0.002
NR-AR-LBD(Androgen receptor) 0.003
NR-Aromatase 0.003
NR-ER(Estrogen receptor) 0.148
NR-ER-LBD(Estrogen receptor) 0.021

Allergy
Skin Sensitization Rule 0
Skin Sensitization 0.115

Acute Toxicity
Acute Toxicity Rule 1
Rat Oral Acute Toxicity 0.422

Organ Toxicity
hERG Blockers 0.003
H-HT(The human hepatotoxicity) 0.013
DILI(Drug-induced liver injury) 0.049

Primary Irritation
Eye Corrosion 0.975
Eye Irritation 0.995
Respiratory Toxicity 0.076

Mutagenic Effects
AMES Toxicity 0.231

Tumorigenic Effects
Carcinogencity 0.111
SR-ARE(Antioxidant Response Element) 0.018
SR-ATAD5(ATPase family AAA domain-containing protein 5) 0.006
SR-p53 0.003

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