Ingredient Details :beta-Fenchyl acetate, exo-


TCMI-ID: TCMI04538


Physicochemical Property
Ingredient Name beta-Fenchyl acetate, exo-
Pubchem CID 156660
Iupac name [(1S,2R,4R)-1,3,3-trimethyl-2-bicyclo[2.2.1]heptanyl] acetate
Molecular Formula C12H20O2
Molecular Weight 196.29
Isomeric smiles CC(=O)O[C@@H]1[C@]2(CC[C@H](C2)C1(C)C)C
InChI InChI=1S/C12H20O2/c1-8(13)14-10-11(2,3)9-5-6-12(10,4)7-9/h9-10H,5-7H2,1-4H3/t9-,10+,12+/m1/s1
InChIKey JUWUWIGZUVEFQB-SCVCMEIPSA-N
External Database Links HERB2.0: HBIN018119   SymMap: SMIT04739   TCMSID: 2459   TCMSP: 2520  
Structural Information
nHA(Number of hydrogen bond acceptors) 2
nHD(Number of hydrogen bond donors) 0
nRot(Number of rotatable bonds) 2
nRing(Number of rings) 2
MaxRing(Number of atoms in the biggest ring) 6
nHet(Number of heteroatoms) 2

Stability
nRig(Number of rigid bonds) 9
Flexibility 0.222
Stereo Centers(Number of stereocenters) 3

Solubility
TPSA(Topological polar surface area) 26.3
logS(The logarithm of aqueous solubility value) -2.822
logP(The logarithm of the n-octanol/water distribution coefficient) 3.159
logD7.4(The logarithm of the n-octanol/water distribution coefficients at pH=7.4) 3.25

Pharmacokinetic Property
Quantitative Estimate of Drug-likeness 0.603
Synthetic accessibility score 4.326
Natural Product-likeness score 2.51
Lipinski Rule Accepted
GSK Rule Accepted
Golden Triangle Rejected

Absorption
Caco-2 Permeability -4.679
MDCK Permeability 2.73E-05
Pgp-substrate 0
HIA(human intestinal absorption) 0.004
F20%(20% Oral Bioavailability) 0.011
F30%(30% Oral Bioavailability) 0.44

Distribution
PPB(Plasma protein binding) 71.90%
VD(Volume Distribution) 1.103
BBB Penetration(Blood brain barrier penetration) 0.213
B3 Penetration(Blood brain barrier penetration) Permeable
Fu(The fraction unbound in plasms) 46.44%

Metabolism
CYP1A2 inhibitor 0.495
CYP1A2 substrate 0.422
CYP2C19 inhibitor 0.231
CYP2C19 substrate 0.839
CYP2C9 inhibitor 0.343
CYP2C9 substrate 0.27
CYP2D6 inhibitor 0.013
CYP2D6 substrate 0.277
CYP3A4 inhibitor 0.119
CYP3A4 substrate 0.314

Excretion
CL(The clearance of a drug) 3.074
T1/2 0.359

Toxicology
NonBiodegradable Rule 0
Pfizer Rule Rejected
SR-MMP 0.029

Toxic Dose
FDAMDD(FDA Maximum (Recommended) Daily Dose) 0.612
IGC50 3.978
LC50FM 5.33
LC50DM 5.541

Reproductive Effects
NR-AR(Androgen receptor) 0.619
NR-AR-LBD(Androgen receptor) 0.009
NR-Aromatase 0.011
NR-ER(Estrogen receptor) 0.07
NR-ER-LBD(Estrogen receptor) 0.019

Allergy
Skin Sensitization Rule 0
Skin Sensitization 0.593

Acute Toxicity
Acute Toxicity Rule 0
Rat Oral Acute Toxicity 0.028

Organ Toxicity
hERG Blockers 0.011
H-HT(The human hepatotoxicity) 0.421
DILI(Drug-induced liver injury) 0.294

Primary Irritation
Eye Corrosion 0.932
Eye Irritation 0.98
Respiratory Toxicity 0.841

Mutagenic Effects
AMES Toxicity 0.021

Tumorigenic Effects
Carcinogencity 0.04
SR-ARE(Antioxidant Response Element) 0.02
SR-ATAD5(ATPase family AAA domain-containing protein 5) 0.005
SR-p53 0.023

Related TCM-Disorder Names

Related Formulae

Related Herbs

Related Targets

Network Analysis

Copyright © Chengdu University of TCM All rights reserved.