Ingredient Details :1,2-Epoxynonadecane


TCMI-ID: TCMI03890


Physicochemical Property
Ingredient Name 1,2-Epoxynonadecane
Pubchem CID 105846
Iupac name 2-heptadecyloxirane
Molecular Formula C19H38O
Molecular Weight 282.5
Isomeric smiles CCCCCCCCCCCCCCCCCC1CO1
InChI InChI=1S/C19H38O/c1-2-3-4-5-6-7-8-9-10-11-12-13-14-15-16-17-19-18-20-19/h19H,2-18H2,1H3
InChIKey CEUXMUYHMURJFZ-UHFFFAOYSA-N
External Database Links HERB2.0: HBIN038441   SymMap: SMIT05191   TCMSID: 2977  
Structural Information
nHA(Number of hydrogen bond acceptors) 1
nHD(Number of hydrogen bond donors) 0
nRot(Number of rotatable bonds) 16
nRing(Number of rings) 1
MaxRing(Number of atoms in the biggest ring) 3
nHet(Number of heteroatoms) 1

Stability
nRig(Number of rigid bonds) 3
Flexibility 5.333
Stereo Centers(Number of stereocenters) 1

Solubility
TPSA(Topological polar surface area) 12.53
logS(The logarithm of aqueous solubility value) -6.911
logP(The logarithm of the n-octanol/water distribution coefficient) 8.185
logD7.4(The logarithm of the n-octanol/water distribution coefficients at pH=7.4) 4.489

Pharmacokinetic Property
Quantitative Estimate of Drug-likeness 0.228
Synthetic accessibility score 2.361
Natural Product-likeness score 0.554
Lipinski Rule Accepted
GSK Rule Rejected
Golden Triangle Accepted

Absorption
Caco-2 Permeability -4.859
MDCK Permeability 1.32E-05
Pgp-substrate 0
HIA(human intestinal absorption) 0.002
F20%(20% Oral Bioavailability) 0.198
F30%(30% Oral Bioavailability) 0.979

Distribution
PPB(Plasma protein binding) 98.13%
VD(Volume Distribution) 1.929
BBB Penetration(Blood brain barrier penetration) 0.064
B3 Penetration(Blood brain barrier penetration) Permeable
Fu(The fraction unbound in plasms) 1.56%

Metabolism
CYP1A2 inhibitor 0.154
CYP1A2 substrate 0.196
CYP2C19 inhibitor 0.263
CYP2C19 substrate 0.062
CYP2C9 inhibitor 0.075
CYP2C9 substrate 0.85
CYP2D6 inhibitor 0.181
CYP2D6 substrate 0.062
CYP3A4 inhibitor 0.185
CYP3A4 substrate 0.045

Excretion
CL(The clearance of a drug) 4.227
T1/2 0.059

Toxicology
NonBiodegradable Rule 2
Pfizer Rule Rejected
SR-MMP 0.114

Toxic Dose
FDAMDD(FDA Maximum (Recommended) Daily Dose) 0.051
IGC50 5.788
LC50FM 5.247
LC50DM 5.669

Reproductive Effects
NR-AR(Androgen receptor) 0.047
NR-AR-LBD(Androgen receptor) 0.002
NR-Aromatase 0.541
NR-ER(Estrogen receptor) 0.327
NR-ER-LBD(Estrogen receptor) 0.029

Allergy
Skin Sensitization Rule 1
Skin Sensitization 0.971

Acute Toxicity
Acute Toxicity Rule 2
Rat Oral Acute Toxicity 0.017

Organ Toxicity
hERG Blockers 0.345
H-HT(The human hepatotoxicity) 0.031
DILI(Drug-induced liver injury) 0.352

Primary Irritation
Eye Corrosion 0.991
Eye Irritation 0.988
Respiratory Toxicity 0.644

Mutagenic Effects
AMES Toxicity 0.016

Tumorigenic Effects
Carcinogencity 0.062
SR-ARE(Antioxidant Response Element) 0.17
SR-ATAD5(ATPase family AAA domain-containing protein 5) 0.004
SR-p53 0.055

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